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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T9419 | Fesoterodine | (R) Fesoterodine | AChR |
Fesoterodine ((R) Fesoterodine) is an orally active, competitive mAChR antagonist with pKi values of 8.0, 7.7, 7.4, 7.3, 7.5 for M1, M2, M3, M4, M5 receptors, respectively. It is used for the overactive bladder (OAB). | |||
T6364 | Desfesoterodine | 5-HMT,(R)-5-Hydroxymethyl Tolterodine,PNU-200577,5-HM,5-hydroxymethyl Tolterodine | AChR |
Desfesoterodine (5-HMT) is a new muscarinic receptor antagonist with Kb of 0.84 nM. |